| Inhibition of the glucose transporter SGLT2 with dapagliflozin in pancreatic alpha cells triggers glucagon secretion C Bonner, J Kerr-Conte, V Gmyr, G Queniat, E Moerman, J Thévenet, ... Nature medicine 21 (5), 512, 2015 | 359 | 2015 |
| Tuberculosis: the drug development pipeline at a glance B Villemagne, C Crauste, M Flipo, AR Baulard, B Déprez, N Willand European journal of medicinal chemistry 51, 1-16, 2012 | 214 | 2012 |
| The bile acid chenodeoxycholic acid increases human brown adipose tissue activity EPM Broeders, EBM Nascimento, B Havekes, B Brans, KHM Roumans, ... Cell metabolism 22 (3), 418-426, 2015 | 160 | 2015 |
| Parallel synthesis of 1, 2, 4-oxadiazoles from carboxylic acids using an improved, uronium-based, activation RF Poulain, AL Tartar, BP Déprez Tetrahedron Letters 42 (8), 1495-1498, 2001 | 151 | 2001 |
| Synthetic EthR inhibitors boost antituberculous activity of ethionamide N Willand, B Dirié, X Carette, P Bifani, A Singhal, M Desroses, F Leroux, ... Nature medicine 15 (5), 537, 2009 | 142 | 2009 |
| Immunization of mice with lipopeptides bypasses the prerequisite for adjuvant. Immune response of BALB/c mice to human immunodeficiency virus envelope glycoprotein. F Martinon, H Gras-Masse, C Boutillon, F Chirat, B Deprez, JG Guillet, ... The Journal of Immunology 149 (10), 3416-3422, 1992 | 128 | 1992 |
| Versatile acylation of N-nucleophiles using a new polymer-supported 1-hydroxybenzotriazole derivative IE Pop, BP Déprez, AL Tartar The Journal of organic chemistry 62 (8), 2594-2603, 1997 | 123 | 1997 |
| Orthogonal combinatorial chemical libraries B Deprez, X Williard, L Bourel, H Coste, F Hyafil, A Tartar Journal of the American Chemical Society 117 (19), 5405-5406, 1995 | 115 | 1995 |
| Efficient propylphosphonic anhydride (® T3P) mediated synthesis of benzothiazoles, benzoxazoles and benzimidazoles X Wen, J El Bakali, R Deprez-Poulain, B Deprez Tetrahedron Letters 53 (19), 2440-2443, 2012 | 105 | 2012 |
| Designing focused chemical libraries enriched in protein-protein interaction inhibitors using machine-learning methods C Reynès, H Host, AC Camproux, G Laconde, F Leroux, A Mazars, ... PLoS computational biology 6 (3), e1000695, 2010 | 103 | 2010 |
| Natural compounds: leads or ideas? Bioinspired molecules for drug discovery T Beghyn, R Deprez‐Poulain, N Willand, B Folleas, B Deprez Chemical biology & drug design 72 (1), 3-15, 2008 | 94 | 2008 |
| Hydroxamates: relationships between structure and plasma stability M Flipo, J Charton, A Hocine, S Dassonneville, B Deprez, ... Journal of medicinal chemistry 52 (21), 6790-6802, 2009 | 86 | 2009 |
| Monitoring of a three-step solid phase synthesis involving a Heck reaction using magic angle spinning NMR spectroscopy IE Pop, CF Dhalluin, BP Déprez, PC Melnyk, GM Lippens, AL Tartar Tetrahedron 52 (37), 12209-12222, 1996 | 86 | 1996 |
| Parallel synthesis of polysubstituted tetrahydroquinolines R Baudelle, P Melnyk, B Déprez, A Tartar Tetrahedron 54 (16), 4125-4140, 1998 | 82 | 1998 |
| Rescue of nonsense mutations by amlexanox in human cells S Gonzalez-Hilarion, T Beghyn, J Jia, N Debreuck, G Berte, K Mamchaoui, ... Orphanet journal of rare diseases 7 (1), 58, 2012 | 81 | 2012 |
| Daytime variation of perioperative myocardial injury in cardiac surgery and its prevention by Rev-Erbα antagonism: a single-centre propensity-matched cohort study and a … D Montaigne, X Marechal, T Modine, A Coisne, S Mouton, G Fayad, ... The Lancet 391 (10115), 59-69, 2018 | 79 | 2018 |
| Comparative efficiency of simple lipopeptide constructs for in vivo induction of virus-specific CTL B Deprez, JP Sauzet, C Boutillon, F Martinon, A Tartar, C Sergheraert, ... Vaccine 14 (5), 375-382, 1996 | 79 | 1996 |
| Ethionamide boosters: synthesis, biological activity, and structure− activity relationships of a series of 1, 2, 4-oxadiazole EthR inhibitors M Flipo, M Desroses, N Lecat-Guillet, B Dirié, X Carette, F Leroux, ... Journal of medicinal chemistry 54 (8), 2994-3010, 2011 | 74 | 2011 |
| Long-lasting anti-viral cytotoxic T lymphocytes induced in vivo with chimeric-multirestricted lipopeptides JP Sauzet, B Déprez, F Martinon, JG Guillet, H Gras-Masse, E Gomard Vaccine 13 (14), 1339-1345, 1995 | 71 | 1995 |
| In silico-in vitro screening of protein-protein interactions: towards the next generation of therapeutics BO Villoutreix, K Bastard, O Sperandio, R Fahraeus, JL Poyet, F Calvo, ... Current pharmaceutical biotechnology 9 (2), 103-122, 2008 | 69 | 2008 |
Bart StaelsProfesseur Université LilleVerified email at pasteur-lille.fr
